Isotonitazepyne

Isotonitazepyne
Identifiers
IUPAC name
  • 5-nitro-2-[4-(2-propoxy)benzyl]-1-[2-(pyrrolidin-1-yl)ethyl]-1H-benzo[d]imidazole
CAS Number
PubChem CID
ChemSpider
Chemical and physical data
FormulaC23H28N4O3
Molar mass408.502 g·mol−1
3D model (JSmol)
SMILES
  • CC(C)OC1=CC=C(C=C1)CC2=NC3=C(N2CCN4CCCC4)C=CC(=C3)[N+](=O)[O-]
InChI
  • InChI=1S/C23H28N4O3/c1-17(2)30-20-8-5-18(6-9-20)15-23-24-21-16-19(27(28)29)7-10-22(21)26(23)14-13-25-11-3-4-12-25/h5-10,16-17H,3-4,11-15H2,1-2H3
  • Key:VRKDSDBBRNHHCR-UHFFFAOYSA-N

Isotonitazepyne (N-pyrrolidino isotonitazene) is a benzimidazole derivative with potent opioid effects, which has been sold as a designer drug over the internet. It has since been identified by the drug checking service CanTEST, in Canberra Australia, and tentatively in New Zealand.[1] It's in vitro potency is approximately 1000 times that of morphine.[2] It is specifically listed as an illegal drug in the US state of Virginia.[3]

See also

References

  1. ↑ "N-pyrrolidino isotonitazene found in counterfeit oxycodone pill r". CanTEST. 9 September 2024. Archived from the original on 9 September 2024. Retrieved 9 September 2024 – via Instagram.
  2. ↑ De Vrieze LM, Walton SE, Pottie E, Papsun D, Logan BK, Krotulski AJ, et al. (September 2024). "In vitro structure-activity relationships and forensic case series of emerging 2-benzylbenzimidazole 'nitazene' opioids". Archives of Toxicology. 98 (9): 2999–3018. doi:10.1007/s00204-024-03774-7. PMC 11324687. PMID 38877156.
  3. ↑ "18VAC110-20-322. Placement of chemicals in Schedule I." Code of Virginia. 2023.
This article is issued from Wikipedia. The text is licensed under Creative Commons - Attribution - Sharealike. Additional terms may apply for the media files.